TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Burnham Institute For Medical Research
Curated by ChEMBL
Burnham Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 269nMAssay Description:Agonist activity against human alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataEC50: 271nMAssay Description:Agonist activity at human alpha4beta2 ACHR expressed in HEK293 cells assessed as change in intracellular calcium concentration by FLIPRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Burnham Institute For Medical Research
Curated by ChEMBL
Burnham Institute For Medical Research
Curated by ChEMBL
Affinity DataEC50: 4.07E+3nMAssay Description:Agonist activity against human alpha3beta4 nAChRMore data for this Ligand-Target Pair