TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 6nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at human thrombopoietin receptor expressed in mouse Ba/F3 cells by kinase activation based reporter gene assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at human thrombopoietin receptor expressed in mouse Ba/F3 cells by kinase activation based reporter gene assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at human thrombopoietin receptor expressed in mouse Ba/F3 cells by kinase activation based reporter gene assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at human thrombopoietin receptor in Ba/F3 cells assessed as activation of Stat5 response element-driven reporter gene expressionMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at TPO receptorMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at TPO receptorMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human TPO receptor expressed in rat BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at TPO receptorMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at human thrombopoietin receptor in Ba/F3 cells assessed as activation of Stat5 response element-driven reporter gene expressionMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at human thrombopoietin receptor expressed in mouse Ba/F3 cells by kinase activation based reporter gene assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at human thrombopoietin receptor in Ba/F3 cells assessed as activation of Stat5 response element-driven reporter gene expressionMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at human thrombopoietin receptor expressed in mouse Ba/F3 cells by kinase activation based reporter gene assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at human thrombopoietin receptor in Ba/F3 cells assessed as activation of Stat5 response element-driven reporter gene expressionMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human thrombopoietin receptor in Ba/F3 cells assessed as activation of Stat5 response element-driven reporter gene expressionMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Agonist activity at human recombinant TPO receptor expressed in mouse BaF3 cells after 24 hrsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Inhibition of human TPOR expressed in human BaF3 cellsMore data for this Ligand-Target Pair
TargetThrombopoietin receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Shanghai Hengrui Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human thrombopoietin receptor transfected in mouse BAF3 cells assessed as stimulation of beta lactamase activity incubated in dar...More data for this Ligand-Target Pair