Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 198120
TargetHistone deacetylase 6 [440-798](Danio rerio)
University of Pennsylvania

LigandPNGBDBM198120(TSA)
Affinity DataKi:  0.800nM ΔG°:  -51.9kJ/mole IC50:  1.40nMT: 2°CAssay Description:The fluorescence anisotropy assay was performed with fluorescein-labeled SAHA (fl-SAHA, gift of C. Fierke, University of Michigan) and measured using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6 [84-835](Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM198120(TSA)
Affinity DataKi:  2.20nM ΔG°:  -49.4kJ/mole IC50:  3.90nMT: 2°CAssay Description:The fluorescence anisotropy assay was performed with fluorescein-labeled SAHA (fl-SAHA, gift of C. Fierke, University of Michigan) and measured using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6 [60-420](Danio rerio)
University of Pennsylvania

LigandPNGBDBM198120(TSA)
Affinity DataKi:  4.80nM ΔG°:  -47.5kJ/mole IC50:  7nMT: 2°CAssay Description:The fluorescence anisotropy assay was performed with fluorescein-labeled SAHA (fl-SAHA, gift of C. Fierke, University of Michigan) and measured using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed