Affinity DataIC50: 1.10nMAssay Description:Activity at human delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro binding affinity towards mu opioid receptors was determined using [3H]-[p-Cl-Phe]- 4] DPDPE or [3H]-Deltorphin IIMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Agonistic efficacy at human delta opioid receptor by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:In vitro binding affinity towards Opioid receptor delta 1 was determined using [3H]-DAMGO or [3H]-CTOPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of DOR in ICR mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction after 3 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Activity at delta opioid receptor in ICR mouse by MVD assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at delta opioid receptor by inhibition of muscle contraction in electrically stimulated isolated mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Agonistic efficacy at rat mu opioid receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:In vitro agonist activity against Opioid receptor mu in guinea pig ileum/longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Activity at mu opioid receptor assessed as contraction of electrically-stimulated Hartley guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Activity at mu opioid receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum longitudinal muscle myenteric plexus assessed as inhibition of electrically-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum longitudinal muscle with myenteric plexus assessed as inhibition of electrically-s...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of mu opioid receptor in guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of electrically-stimulated musc...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of MOR in Hartley guinea pig ileum longitudinal muscle myenteric plexus assessed as inhibition of electrically-stimulated muscle contracti...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor by inhibition of muscle contraction in electrically stimulated isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-induced smooth muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:In vitro agonist activity against Opioid receptor delta in mouse vas deferensMore data for this Ligand-Target Pair