TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences
Curated by ChEMBL
Wuhan University School of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair