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Found 3 of ic50 for monomerid = 50420675
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50420675(CHEMBL2087059)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat TRPM8 expressed in HEK293 cells assessed as reduction in 20 uM menthol-stimulated increase in intracellular Ca2+ levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50420675(CHEMBL2087059)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat TRPM8 expressed in HEK293 cells assessed as reduction in 0.25 uM icilin-stimulated increase in intracellular Ca2+ levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50420675(CHEMBL2087059)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of rat TRPA1 expressed in HEK293 cells assessed as reduction in 100 uM allyl isothiocyanate-stimulated increase in intracellular Ca2+ leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed