Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50051291
TargetNeuromedin-K receptor(Homo sapiens (Human))
Smithkline Beecham

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards cloned human Tachykinin receptor 3 (hNK-3) expressed in CHO cells using [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Smithkline Beecham

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  31nMAssay Description:Inhibition of [125I]-MePhe7-Neurokinin B (NKB) binding in human Tachykinin receptor 3 of chinese hamster ovary (hNK-3-CHO) cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Smithkline Beecham

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  31nMAssay Description:Binding Affinity of [125I]-MePhe7-NKB towards Tachykinin receptor 3-CHO cell membranes(n=3-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Smithkline Beecham

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  31.6nMAssay Description:Binding affinity to human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Smithkline Beecham S.P.A. Milano

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  2.95E+3nMAssay Description:Inhibition of [125I]-Neurokinin A (NKA) binding in human Tachykinin receptor 2 of chinese hamster ovary (hNK-2-CHO) cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Smithkline Beecham S.P.A. Milano

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi:  2.95E+3nMAssay Description:Binding Affinity of [125I]NKA towards Tachykinin receptor 2-CHO cell membranes (n=3-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Smithkline Beecham S.P.A. Milano

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-substance P binding in human Tachykinin receptor 1 of chinese hamster ovary (hNK-1-CHO) cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Smithkline Beecham S.P.A. Milano

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding Affinity of [3H]- substance P towards Tachykinin receptor 1-CHO cell membranes (n=3-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed