Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ki for monomerid = 50244036
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha1beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  15nMAssay Description:Binding affinity to human recombinant GABAA alpha2 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha2beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  18.9nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha3beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human recombinant GABAA alpha3 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  110nMAssay Description:Binding affinity to human recombinant GABAA alpha5 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha5beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  897nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha4beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human recombinant GABAA alpha4 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  4.75E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human recombinant GABAA alpha6 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]flunitrazepam from human recombinant GABAA alpha6beta3gamma2 receptor expressed in HEK cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed