Affinity DataKi: 25nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.39E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced ethidium uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 4.42E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in SK-N-MC cells assessed as inhibition of forskolin-stimulated cAMP accumulation treate...More data for this Ligand-Target Pair