Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50408804
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50408804(CHEMBL5290025)
Affinity DataKi:  25nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
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TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50408804(CHEMBL5290025)
Affinity DataKi:  4.39E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced ethidium uptakeMore data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50408804(CHEMBL5290025)
Affinity DataKi:  4.42E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in SK-N-MC cells assessed as inhibition of forskolin-stimulated cAMP accumulation treate...More data for this Ligand-Target Pair
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