Affinity DataKd: 7.20nMAssay Description:Binding affinity to human DYRK1A assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.80nMAssay Description:Binding affinity to DYRK1AMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Binding affinity to CLK4More data for this Ligand-Target Pair
Affinity DataKd: 75nMAssay Description:Binding affinity to CLK1More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to DYRK1BMore data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Binding affinity to HIPK3More data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding affinity to HIPK1More data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Binding affinity to CLK2More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataKd: 450nMAssay Description:Binding affinity to DYRK2More data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding affinity to GSK3AMore data for this Ligand-Target Pair
Affinity DataKd: 561nMAssay Description:Binding affinity to human GSK-3beta assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 930nMAssay Description:Binding affinity to IRAK1More data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to CLK3More data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to TAOK1More data for this Ligand-Target Pair