Compile Data Set for Download or QSAR
maximum 50k data
Found 15 of kd for monomerid = 50347750
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  7.20nMAssay Description:Binding affinity to human DYRK1A assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  7.80nMAssay Description:Binding affinity to DYRK1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  8.5nMAssay Description:Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  70nMAssay Description:Binding affinity to CLK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  75nMAssay Description:Binding affinity to CLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  140nMAssay Description:Binding affinity to DYRK1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  230nMAssay Description:Binding affinity to HIPK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  320nMAssay Description:Binding affinity to HIPK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  360nMAssay Description:Binding affinity to CLK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  450nMAssay Description:Binding affinity to DYRK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  550nMAssay Description:Binding affinity to GSK3AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  561nMAssay Description:Binding affinity to human GSK-3beta assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  930nMAssay Description:Binding affinity to IRAK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to CLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to TAOK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed