Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50002172
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454561(CHEMBL4214185)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454561(CHEMBL4214185)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454558(CHEMBL4217119)
Affinity DataKi:  4.39E+3nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454560(CHEMBL4218602)
Affinity DataKi:  7.89E+3nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454564(CHEMBL4209269)
Affinity DataKi:  1.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454554(CHEMBL4209786)
Affinity DataKi:  2.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454564(CHEMBL4209269)
Affinity DataKi:  2.50E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454559(CHEMBL4202934)
Affinity DataKi:  3.35E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454557(CHEMBL4214761)
Affinity DataKi:  3.38E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454554(CHEMBL4209786)
Affinity DataKi:  3.62E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50037773(CHEMBL3358195)
Affinity DataKi:  4.32E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454563(CHEMBL4204907)
Affinity DataKi:  5.23E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454560(CHEMBL4218602)
Affinity DataKi:  7.40E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454565(CHEMBL4210507)
Affinity DataKi:  7.81E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454562(CHEMBL4208846)
Affinity DataKi:  8.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454562(CHEMBL4208846)
Affinity DataKi:  8.38E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454553(CHEMBL4202968)
Affinity DataKi:  9.54E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454558(CHEMBL4217119)
Affinity DataKi:  2.68E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454559(CHEMBL4202934)
Affinity DataKi:  3.65E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50037773(CHEMBL3358195)
Affinity DataKi:  3.73E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454563(CHEMBL4204907)
Affinity DataKi:  3.93E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454565(CHEMBL4210507)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454552(CHEMBL4213668)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454552(CHEMBL4213668)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454553(CHEMBL4202968)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454557(CHEMBL4214761)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed