Affinity DataIC50: 0nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam and testosterone as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of CYP2B6 in human liver microsomes using bupropion as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of hERG expressed in HEK293 cells by automated patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataIC50: 3.71E+3nMAssay Description:Inhibition of hERG expressed in HEK293 cells by automated patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataIC50: 4.91E+3nMAssay Description:Inhibition of hERG expressed in HEK293 cells by automated patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.73E+3nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam and testosterone as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam and testosterone as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2B6 in human liver microsomes using bupropion as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2B6 in human liver microsomes using bupropion as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 2.41E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 510nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 660nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.64E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.61E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 3.52E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.22E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.04E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 420nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Homo sapiens)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
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