Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50018769
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612294(CHEMBL5281395)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612293(CHEMBL5265996)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612290(CHEMBL5288132)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612285(CHEMBL5269564)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612287(CHEMBL5274333)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612292(CHEMBL5268272)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612295(CHEMBL5267547)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612291(CHEMBL5278471)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50514710(CHEMBL4555677)
Affinity DataIC50:  62nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612294(CHEMBL5281395)
Affinity DataIC50:  69nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612289(CHEMBL5282634)
Affinity DataIC50:  110nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612288(CHEMBL5281552)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612286(CHEMBL5287156)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612290(CHEMBL5288132)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612293(CHEMBL5265996)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612285(CHEMBL5269564)
Affinity DataIC50:  410nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612284(CHEMBL5283409)
Affinity DataIC50:  440nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612291(CHEMBL5278471)
Affinity DataIC50:  580nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612295(CHEMBL5267547)
Affinity DataIC50:  630nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612292(CHEMBL5268272)
Affinity DataIC50:  790nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612280(CHEMBL5269301)
Affinity DataIC50:  6.30E+3nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612278(CHEMBL5281757)
Affinity DataIC50:  8.20E+3nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612277(CHEMBL5274695)
Affinity DataIC50:  8.70E+3nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612283(CHEMBL5271896)
Affinity DataIC50:  1.60E+4nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612281(CHEMBL5280443)
Affinity DataIC50:  5.30E+4nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50514710(CHEMBL4555677)
Affinity DataIC50:  5.60E+4nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612296(CHEMBL5284552)
Affinity DataIC50:  5.70E+4nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612276(CHEMBL5272193)
Affinity DataIC50:  6.60E+4nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612279(CHEMBL5273013)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDeoxyhypusine synthase(Homo sapiens)TBA
LigandPNGBDBM50612282(CHEMBL5271847)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]spermidine trihydrochloride from N-terminal 6his tagged TEV fused human DHPS expressed in Escherichia coli BL21 (DE3) incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed