Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50018815
TargetCyclin-dependent kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50612866(CHEMBL5266005)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612866(CHEMBL5266005)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612866(CHEMBL5266005)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612866(CHEMBL5266005)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50013510(CHEMBL3263773)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
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TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM164883(US9067888, 33)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
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TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50511926(CHEMBL4442620)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50516532(CHEMBL4560679)
Affinity DataIC50:  6nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
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TargetCyclin-dependent kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50511926(CHEMBL4442620)
Affinity DataIC50:  7nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
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LigandPNGBDBM50516532(CHEMBL4560679)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50511926(CHEMBL4442620)
Affinity DataIC50:  9nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50612868(CHEMBL5283843)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50193097(CHEMBL3940387)
Affinity DataIC50:  11nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
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TargetCyclin-dependent kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50511926(CHEMBL4442620)
Affinity DataIC50:  11nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
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TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50612869(CHEMBL5270061)
Affinity DataIC50:  27nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  30nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

LigandPNGBDBM50612870(CHEMBL5272692)
Affinity DataIC50:  60nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50612867(CHEMBL5273318)
Affinity DataIC50:  86nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50612871(CHEMBL5272649)
Affinity DataIC50:  86nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using as PDKtide substrate incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  170nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50193097(CHEMBL3940387)
Affinity DataIC50:  400nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50612867(CHEMBL5273318)
Affinity DataIC50:  637nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50612869(CHEMBL5270061)
Affinity DataIC50:  796nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50612868(CHEMBL5283843)
Affinity DataIC50:  876nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50612870(CHEMBL5272692)
Affinity DataIC50:  915nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50612871(CHEMBL5272649)
Affinity DataIC50:  924nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50516532(CHEMBL4560679)
Affinity DataIC50:  975nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) incubated for 1 hr in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50516532(CHEMBL4560679)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50013510(CHEMBL3263773)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM164883(US9067888, 33)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed