Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50019055
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201158(4-(4-hydroxyphenyl)benzo[b]thiophene-7-carbaldehyd...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201160(7-(4-hydroxyphenyl)benzo[b]thiophene-4-carbaldehyd...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201159(4-(3-fluoro-4-hydroxyphenyl)-1-naphthaldehyde oxim...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201164(4-(4-HYDROXYPHENYL)-1-NAPHTHALDEHYDE OXIME | CHEMB...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201161(1-(3-fluoro-4-hydroxyphenyl)-2-methyl-1H-indole-3-...)
Affinity DataIC50:  8.05nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201156(3,5-dichloro-3'-fluoro-4'-hydroxy-biphenyl-4-carba...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  9.70nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201163(4-(4-hydroxyphenyl)benzofuran-7-carbaldehyde oxime...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201155(1-(4-hydroxyphenyl)-2-methyl-1H-indole-3-carbaldeh...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201158(4-(4-hydroxyphenyl)benzo[b]thiophene-7-carbaldehyd...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201160(7-(4-hydroxyphenyl)benzo[b]thiophene-4-carbaldehyd...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201164(4-(4-HYDROXYPHENYL)-1-NAPHTHALDEHYDE OXIME | CHEMB...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201159(4-(3-fluoro-4-hydroxyphenyl)-1-naphthaldehyde oxim...)
Affinity DataIC50:  148nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201163(4-(4-hydroxyphenyl)benzofuran-7-carbaldehyde oxime...)
Affinity DataIC50:  155nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201162(1-(4-hydroxyphenyl)-1H-indole-3-carbaldehyde oxime...)
Affinity DataIC50:  202nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201156(3,5-dichloro-3'-fluoro-4'-hydroxy-biphenyl-4-carba...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201155(1-(4-hydroxyphenyl)-2-methyl-1H-indole-3-carbaldeh...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201161(1-(3-fluoro-4-hydroxyphenyl)-2-methyl-1H-indole-3-...)
Affinity DataIC50:  298nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  395nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201157(7-(4-hydroxyphenyl)benzofuran-4-carbaldehyde oxime...)
Affinity DataIC50:  457nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201157(7-(4-hydroxyphenyl)benzofuran-4-carbaldehyde oxime...)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201162(1-(4-hydroxyphenyl)-1H-indole-3-carbaldehyde oxime...)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed