TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 20.8nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 21.1nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 7.02E+3nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataKi: 1.35E+4nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 21.8nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 28.3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 143nMAssay Description:Inhibition of LPA3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 184nMAssay Description:Inhibition of LPA3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 347nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: >7.30E+3nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: >9.40E+3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 1.39E+4nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 2.74E+4nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataEC50: >1.18E+4nMAssay Description:Agonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataEC50: >1.14E+4nMAssay Description:Agonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataEC50: >1.23E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair