Affinity DataKi: 0.380nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.91nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.83nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 284nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 352nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 442nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 474nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 498nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 519nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 543nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 766nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 838nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 838nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.18E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.19E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.19E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.28E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.02E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.02E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.84E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 4.32E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor kappa 1 on guinea pig cerebellum membranes by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair