Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50039020
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304252((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  6.94nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304253((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  8.51nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304254((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304259((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  16.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304256((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  10.1nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304257((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  75.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304258((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  20.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304255((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  13.2nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed