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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM255474'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM255474(US9481688, 1 | US9481688, 3)
Affinity DataKi:  3.37nM ΔG°:  -48.4kJ/molepH: 7.6 T: 2°CAssay Description:[3H]-Ketanserin binding experiments are carried out in SPA 96-well format. Membranes used in this assay are prepared from AV-12 cells stably expressi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM255474(US9481688, 1 | US9481688, 3)
Affinity DataKi:  7.01nM ΔG°:  -46.5kJ/molepH: 7.6 T: 2°CAssay Description:[3H]-Ketanserin binding experiments are carried out in SPA 96-well format. Membranes used in this assay are prepared from AV-12 cells stably expressi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent