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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50409488'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  13nMAssay Description:In vitro ability to displace [3H]ketanserin binding from 5-hydroxytryptamine 2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  13nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad De Santiago

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed