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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50004589'
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50004589(8-Cyclopentyl-1,3-diethyl-3,7-dihydro-purine-2,6-d...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human recombinant A1 receptor expressed in CHOA1 cell membranes incubated for 60 mins by radioligand binding competiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50004589(8-Cyclopentyl-1,3-diethyl-3,7-dihydro-purine-2,6-d...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human recombinant A1 receptor expressed in CHOA1 cell membranes incubated for 60 mins by radioligand binding competiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50004589(8-Cyclopentyl-1,3-diethyl-3,7-dihydro-purine-2,6-d...)
Affinity DataKi:  19nMAssay Description:Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed