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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50080289'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Cadus Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50080289((R)-3-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyri...)
Affinity DataKi:  962nMAssay Description:Inhibitory activity against binding of [3H]-DPCPX to human A1 receptor (hA1) using competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Cadus Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50080289((R)-3-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyri...)
Affinity DataIC50:  2.06E+3nMAssay Description:Binding affinity towards human A1 receptor (hA1) was measured through displacement of [3H]-DPCPX using mammalian cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Cadus Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50080289((R)-3-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyri...)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibitory activity against binding of [3H]-CGS-21,680 to human A2a receptor (hA2a) using competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed