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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50235050'
TargetAdenosine receptor A2a(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50235050(CHEMBL4099543)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50235050(CHEMBL4099543)
Affinity DataKi:  27nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed