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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1B adrenergic receptor' and Ligand = 'BDBM84440'
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  43nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  54.5nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  225nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed