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Found 3 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50154006'
TargetAndrogen receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50:  0.00900nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed