TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataKd: 145nMAssay Description:Displacement of [3H]-CGP12177 from human beta2 adrenoceptor expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataEC50: 60nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataKd: 85nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataKd: 56nMAssay Description:Antagonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair