Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM35872'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM35872(5,6-bis(4-methoxyphenyl)-N-(piperidin-1-yl)pyrazin...)
Affinity DataIC50:  21nMpH: 7.4 T: 2°CAssay Description:A GTP-gamma-S CB1 functional assay was used to assess the potency of the pyrazine derivatives. [35S]GTP-gamma-S binding assays were performed at 30 d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM35872(5,6-bis(4-methoxyphenyl)-N-(piperidin-1-yl)pyrazin...)
Affinity DataIC50:  42.7nMAssay Description:Antagonist activity against human recombinant cannabinoid-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed