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Found 2 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50329183'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329183(2-(4-benzyl-5-oxo-1-phenyl-4H-benzo[b][1,2,4]triaz...)
Affinity DataIC50:  201nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329183(2-(4-benzyl-5-oxo-1-phenyl-4H-benzo[b][1,2,4]triaz...)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed