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Found 3 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 9' and Ligand = 'BDBM50253621'
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50253621((S)-4-amino-5-((R)-2-boronopyrrolidin-1-yl)-5-oxop...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50253621((S)-4-amino-5-((R)-2-boronopyrrolidin-1-yl)-5-oxop...)
Affinity DataIC50:  13nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50253621((S)-4-amino-5-((R)-2-boronopyrrolidin-1-yl)-5-oxop...)
Affinity DataIC50:  1.30E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
In DepthDetails US Patent