Found 1 Enz. Inhib. hit(s) with Target = 'Disintegrin and metalloproteinase domain-containing protein 17' and Ligand = 'BDBM237181'
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
China Pharmaceutical University
China Pharmaceutical University
Affinity DataIC50: 8.00E+3nMpH: 7.4 T: 2°CAssay Description:TACE was purchased as an active form enzyme (R&D Systems). Hydrolysis of the TACE-substrate Mca-Pro-Leu-Ala-Gln-Ala-Val-Dpa-Arg-Ser-Ser-Ser-Arg-NH (s...More data for this Ligand-Target Pair