Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Disintegrin and metalloproteinase domain-containing protein 17' and Ligand = 'BDBM429761'
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM429761((5R)-5-[3-[4- (4-fluoro-3,5- dimethoxy- phenyl)-1-...)
Affinity DataIC50:  75nMAssay Description:The basis for the assay is the cleavage of the substrate 5FAM-LAQAVRSSSRK-5TAMRA (SEQ ID No 3) (Anaspec, custom 34891) by human TACE (R&D SYSTEMS INC...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent