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Found 2 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor' and Ligand = 'BDBM50192478'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192478(1-(3-bromo-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192478(1-(3-bromo-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed