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Found 4 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50252365'
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252365((R,S)-amino-(1-hydroxy-4-ethyl-pyrazol-3-yl)-aceti...)
Affinity DataEC50:  4.70E+4nMAssay Description:Activity at rat recombinant NR1/NR2A receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252365((R,S)-amino-(1-hydroxy-4-ethyl-pyrazol-3-yl)-aceti...)
Affinity DataEC50:  4.30E+4nMAssay Description:Activity at rat NR1/NR2D receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252365((R,S)-amino-(1-hydroxy-4-ethyl-pyrazol-3-yl)-aceti...)
Affinity DataEC50:  9.10E+4nMAssay Description:Activity at rat recombinant NR1/NR2C receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252365((R,S)-amino-(1-hydroxy-4-ethyl-pyrazol-3-yl)-aceti...)
Affinity DataEC50:  6.80E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed