Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]NAMH from human cloned histamine 3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]NAMH from rat cloned histamine 3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Antagonist activity at human histamine 3 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair