Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50480524'
TargetIntegrase(Human immunodeficiency virus 1)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50480524(CHEMBL562366)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50480524(CHEMBL562366)
Affinity DataIC50:  140nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity expressed in Escherichia coli after 30 mins using [32P]-labeled oligonucleotide as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50480524(CHEMBL562366)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing activity expressed in Escherichia coli after 30 mins using [32P]-labeled oligonucleotide as a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50480524(CHEMBL562366)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed