Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50092699'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50092699(CHEMBL126842 | N,N-Diethyl-4-[(1-methyl-piperidin-...)
Affinity DataIC50: >8.90E+3nMAssay Description:Binding affinity on cloned opioid receptor kappa 1 in human HEK293S cells using [125I]-D-Pro10-dynorphin A[1-11] as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed