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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 5' and Ligand = 'BDBM50243715'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50:  8.27E+4nMAssay Description:Inhibition of ASK1 (unknown origin) by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ASK1 (unknown origin) by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed