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Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM50048580'
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Hoechst-Roussel Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50048580(CHEMBL29835 | Indol-1-yl-propyl-pyridin-4-yl-amine...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against [3H]oxotremorine-M binding to muscarinic receptors in rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Hoechst-Roussel Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50048580(CHEMBL29835 | Indol-1-yl-propyl-pyridin-4-yl-amine...)
Affinity DataIC50:  940nMAssay Description:Inhibition of [3H]quinuclidinyl benzilate (QNB) binding from rat forebrain membranes in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Hoechst-Roussel Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50048580(CHEMBL29835 | Indol-1-yl-propyl-pyridin-4-yl-amine...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [3H]quinuclidinyl benzilate (QNB) binding from rat forebrain membranes in the absence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed