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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50062588'
TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50062588(3-(3-Butoxy-pyrazin-2-yloxy)-1-aza-bicyclo[2.2.2]o...)
Affinity DataIC50:  22.3nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 using [3H]-Pirenzepine (Pz) radioligand in rat hippocampus membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50062588(3-(3-Butoxy-pyrazin-2-yloxy)-1-aza-bicyclo[2.2.2]o...)
Affinity DataIC50:  38nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 using [3H]-oxotremorine-M (Oxo-M) radioligand in rat hippocampus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed