Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50347783'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Heptares Therapeutics
Curated by ChEMBL
Heptares Therapeutics
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at human M1 muscarinic receptor expressed in CHO cells assessed as inhibition of carbachol-stimulated phosphatidyl-inositol hydrolys...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Heptares Therapeutics
Curated by ChEMBL
Heptares Therapeutics
Curated by ChEMBL
Affinity DataEC50: 7.94nMAssay Description:Agonist activity at human muscarinic M1 receptor expressed in CHO cells assessed as intracellular calcium mobilization after 10 to 15 mins by FLIPR a...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Heptares Therapeutics
Curated by ChEMBL
Heptares Therapeutics
Curated by ChEMBL
Affinity DataEC50: 5.01nMAssay Description:Agonist activity at human muscarinic M1 receptor expressed in CHO cells assessed as effect on calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair