Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50004664'
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Ability of the compound to displace [3H]-methylscopolamine ([3H]-NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Mus musculus)
University of South Carolina
Curated by ChEMBL
University of South Carolina
Curated by ChEMBL
Affinity DataKi: 9.50E+3nMAssay Description:Ability of the compound to displace [3H]-methylscopolamine ([3H]-NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Binding affinity of the compound against rat muscarinic acetylcholine receptor M2 using heart tissue and [3H]-N-methylscopolamineMore data for this Ligand-Target Pair