Affinity DataIC50: 96nMAssay Description:Displacement of ([125I]-His3, MePhe7)-NKB from NK3R (unknown origin) transfected in CHO cells by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Activity at human NK3 receptor expressed in CHO cells assessed as increase in inositol phosphate generationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.70nMAssay Description:Activity at human NK3 receptor assessed as stimulation of inositol phosphate generation in CHO cellsMore data for this Ligand-Target Pair