Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50299253'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299253((S)-2-(5-methoxybenzo[d]thiazol-2-ylthio)propanoic...)
Affinity DataEC50:  3.33E+4nMAssay Description:Agonist activity at human PPARalpha expressed in HEK293 cells assessed as receptor transactivation at by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299253((S)-2-(5-methoxybenzo[d]thiazol-2-ylthio)propanoic...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human PPARalpha expressed in HEK293 cells assessed as receptor transactivation at by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed