Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50299264'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50299264(2-[(6-Bromo-1,3-benzothiazol-2-yl)thio]-2-methylpr...)
Affinity DataEC50:  4.58E+4nMAssay Description:Agonist activity at human PPARalpha expressed in HEK293 cells assessed as receptor transactivation at by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed