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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50503119'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503119(CHEMBL4518548)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503119(CHEMBL4518548)
Affinity DataEC50:  4.40nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed