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Found 2 Enz. Inhib. hit(s) with Target = 'Protein kinase C zeta type' and Ligand = 'BDBM50353647'
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed