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Found 2 Enz. Inhib. hit(s) with Target = 'Receptor-interacting serine/threonine-protein kinase 1' and Ligand = 'BDBM50263163'
TargetReceptor-interacting serine/threonine-protein kinase 1(Mus musculus)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50263163(CHEMBL4099814)
Affinity DataIC50:  640nMAssay Description:Inhibition of RIPK1 in mouse L929sA cells transfected with human Fas assessed as inhibition in TNF-induced necroptosis pretreated for 24 hrs followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Mus musculus)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50263163(CHEMBL4099814)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of RIPK1 in mouse L929sA cells transfected with human Fas assessed as inhibition in TNF-induced necroptosis pretreated for 24 hrs followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed