Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor gamma' and Ligand = 'BDBM50132580'
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50132580((2E,4E,6E)-7-[3,5-Di-tert-butyl-2-(2,2-difluoro-et...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against RAR gamma receptor using [3H]-ATRA as radioligand in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50132580((2E,4E,6E)-7-[3,5-Di-tert-butyl-2-(2,2-difluoro-et...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed