Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase haspin' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Gachon University
Curated by ChEMBL
Gachon University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Gachon University
Curated by ChEMBL
Gachon University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Gachon University
Curated by ChEMBL
Gachon University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Gachon University
Curated by ChEMBL
Gachon University
Curated by ChEMBL
Affinity DataIC50: 75.6nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair