Found 1 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM50510173'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Spanish National Cancer Research Centre (Cnio)
Curated by ChEMBL
Spanish National Cancer Research Centre (Cnio)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of PIM1 (unknown origin) using PIM2tide as substrate in presence of [gamma-33P]ATP incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair